SB1317 hydrochloride

CAS No.

SB1317 hydrochloride ( TG-02 hydrochloride )

Catalog No. M19398 CAS No.

SB1317 is an effective inhibitor of CDK2/JAK2/FLT3 (IC50: 13/73/56 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 70 Get Quote
5MG 125 Get Quote
10MG 206 Get Quote
25MG 370 Get Quote
50MG 451 Get Quote
100MG Get Quote Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    SB1317 hydrochloride
  • Note
    Research use only not for human use.
  • Brief Description
    SB1317 is an effective inhibitor of CDK2/JAK2/FLT3 (IC50: 13/73/56 nM).
  • Description
    SB1317 is an effective inhibitor of CDK2/JAK2/FLT3 (IC50: 13/73/56 nM).
  • Synonyms
    TG-02 hydrochloride
  • Pathway
    Angiogenesis
  • Target
    CDK
  • Recptor
    CDK2; FLT3; JAK2
  • Research Area
    Cancer
  • Indication
    Anaplastic astrocytoma; Glioblastoma

Chemical Information

  • CAS Number
    --
  • Formula Weight
    408.92
  • Molecular Formula
    C23H25ClN4O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:26.5 mg/mL
  • SMILES
    Cl.CN1C\C=C\CCOc2cccc(c2)-c2ccnc(Nc3cccc(C1)c3)n2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.William AD et al. Discovery of kinase spectrum selective macrocycle (16E)-14-methyl-20-oxa-571426-tetraazatetracyclo[19.3.1.1(26).1(812)]heptacosa-1(25)2(26)358(27)911162123-decaene (SB1317/TG02) a potent inhibitor of cyclin dependent kina.
molnova catalog
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